tcsc7421 Benzquinamide

Benzquinamide (P2647) is an antiemetic which can bind to the α_2A, α_2B, and α_2C adrenergic receptors (α2-AR) with K_i values of 1,365, 691, and 545 nM, respectively.

IC50 & Target: K_i: 1,365 nM (α_2A), 691 nM (α_2B), 545 nM (α_2C)^[1].