tcsc2236 NVP-QAV-572

NVP-QAV-572 is a PI3K inhibitor extracted from patent US7998990B2, Compound Example 8, has an IC₅₀ of 10 nM.

IC50 & Target: IC50: 10 nM (PI3K)^[1]

In Vitro: NVP-QAV-572 (Example 8) is useful in the treatment of conditions which are mediated by the activation of the Pi3 kinase enzymes, particularly inflammatory or allergic conditions^[1].