tcsc1000 VU 0364439

Order Now

AVAILABLE SIZES

$189.00 ORDERING INFORMATION International
TAICLONE BIOTECH CORP.
order@taiclone.com
+886-2-2735-9682
+886-2-2735-9807

Data sheet

Download PDF Datasheet

Technical Inquries

Submit Review

Product Description

VU 0364439 is a mGlu4 positive allosteric modulator (PAM), with EC50 of 19.8 nM.

IC50 Value: 19.8 nM(EC50)

Target: mGluR

in vitro:

in vivo: VU 0364439 possess less than ideal PK properties preventing their use as in vivo tools. It shows better stability in HLM (63% remaining) than RLM (2% remaining).

Information

CAS No1246086-78-1
FormulaC18H13Cl2N3O3S
Clinical Informationclinicalinformation
PathwayGPCR/G Protein
TargetmGluR

Specifications

Purity / Grade>98%
SolubilityDMSO : 50 mg/mL (118.40 mM; Need ultrasonic)
Smilessmiles

Misc Information

Observed Molecular Weight422.29
Get valuable resources and offers directly to your email.