tcsc0018479 CB2R-IN-1

CB2R-IN-1 is a potent cannabinoid CB₂ receptor inverse agonist with a K_i of 0.9 nM.

IC50 & Target: Ki: 0.9 nM (Cannabinoid CB₂ receptor)^[1]

In Vitro: CB2R-IN-1 (Compound 37) is a potent cannabinoid CB₂ receptor ligand (K_i=0.9 nM) with excellent selectivity over the CB₁ receptor (K_i=8259.3 nM)^[1].