tcsc0018471 AVE5688

AVE5688 is an inhibitor of glycogen phosphorylase (GP), with IC₅₀s of 430 nM and 915 nM and K_ds of 170 nM and 530 nM for rabbit muscle glycogen phosphorylase (rmGPb and rmGPa, respectively); AVE5688 can be used for the research of type 2 diabetes.

IC50 & Target: IC50: 430 nM (rmGPb), 915 nM (rmGPa)^[1]


Kd: 170 nM (rmGPb), 530 nM (rmGPa)^[1]

In Vitro: AVE5688 is an inhibitor of glycogen phosphorylase (GP), with IC₅₀s of 430 nM and 915 nM and K_ds of 170 nM and 530 nM for rabbit muscle glycogen phosphorylase (rmGPb and rmGPa, respectively)^[1].