tcsc2102 Mutant IDH1 inhibitor

Mutant IDH1 inhibitor is a potent mutant IDH1 R132H inhibitor with IC₅₀ of < 72 nM.

IC50 & Target: IC50: < 72 nM (mutant IDH1 R132H)

In Vitro: Mutant IDH1 inhibitor is a potent IDH1 R132H inhibitor, and used for the treatment of diseases or disorders associated with such mutant IDH proteins including, but not limited to, cell-proliferation disorders, such as cancer^[1].