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BioChemicals
GSK2606414
tcsc1428
GSK2606414
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AVAILABLE SIZES
5mg
10mg
50mg
100mg
200mg
$
170.00
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ORDERING INFORMATION
International
TAICLONE BIOTECH CORP.
order@taiclone.com
+886-2-2735-9682
+886-2-2735-9807
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Western blot (WB)
Immunohistochemistry (IHC)
Immunofluorescence (IF)
Immunocytochemistry (ICC)
Immunoprecipitation (IP)
Co-Immunoprecipitation (CoIP)
Chromatin Immunoprecipitation (ChIP)
RNA Binding Protein Immunoprecipitation (RIP)
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Product Description
GSK2606414 is an orally available and selective
PERK
inhibitor with an
IC
50
of 0.4 nM.
IC50 & Target: IC50: 0.4 nM (PERK)
In Vitro:
GSK2606414 inhibits PERK activation in cells
[1]
.
In Vivo:
GSK2606414 (50 and 150 mg/kg, p.o.) inhibits the growth of a human tumor xenograft in mice
[1]
.
Information
CAS No
1337531-36-8
Formula
C
24
H
20
F
3
N
5
O
Clinical Information
clinicalinformation
Pathway
Cell Cycle/DNA Damage
Target
PERK
Specifications
Purity / Grade
>98%
Solubility
DMSO : ≥ 31 mg/mL (68.67 mM)
Smiles
smiles
Misc Information
Observed Molecular Weight
451.44
related data
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