tcsc0913 LY2183240

Order Now

AVAILABLE SIZES

$114.00 ORDERING INFORMATION International
TAICLONE BIOTECH CORP.
order@taiclone.com
+886-2-2735-9682
+886-2-2735-9807

Data sheet

Download PDF Datasheet

Technical Inquries

Submit Review

Product Description

LY2183240 is a novel and highly potent blocker of anandamide uptake (IC50 = 270 pM). LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM).

IC50: 270 pM (anandamide uptake); 12.4 nM (FAAH)

Target: FAAH; Anandamide uptake

Following i.p. administration in rats, LY2183240 increases brain anandamide concentration and exerts antinociceptive effects in formalin model of pain.

Information

CAS No874902-19-9
FormulaC17H17N5O
Clinical Informationclinicalinformation
PathwayNeuronal Signaling
Metabolic Enzyme/Protease
TargetFAAH
FAAH

Specifications

Purity / Grade>98%
SolubilityDMSO : 50 mg/mL (162.68 mM; Need ultrasonic)
Smilessmiles

Misc Information

Observed Molecular Weight307.35
Get valuable resources and offers directly to your email.