tcsc0889 (R) -Baclofen

(R)-Baclofen(STX209) is a selective GABAB receptor agonist. IC50 value:

Target: GABAB receptor

GABAB receptors are metabotropic receptors which produce slow inhibitory signals. By manipulating GABAB receptor activity using Baclofen, a variety of functions are studied including synaptic transmissions and antinociception events.