tcsc0016966 Tilapertin

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Product Description

Tilapertin is an oral inhibitor of glycine transporter type-1 (GlyT1).

IC50 & Target: GlyT1[1]

In Vivo: Tilapertin is a nanomolar potent, orally bioavailable and selective GlyT1 inhibitor. Oral administration of Tilapertin dose-dependently increases cerebrospinal fluid (CSF) glycine concentration in rats[1].

Information

CAS No1000690-85-6
FormulaC20H21F3N2O2
Clinical Informationclinicalinformation
PathwayNeuronal Signaling
Membrane Transporter/Ion Channel
TargetGlyT
GlyT

Specifications

Purity / Grade>98%
Solubility10 mM in DMSO
Smilessmiles

Misc Information

Alternative NamesAMG747
Observed Molecular Weight378.39
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